SCHEMBL19003474

SCHEMBL19003474

OC(/C=C/c1ccc(-c2ccccc2)s1)Nc1ccc(-n2ccnc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
KMT2A Q03164 1/20 0.47
PORCN Q9H237 8/20 0.45
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.40
ACP1 P24666 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
ADH5 P11766 1/20 0.38
ENPP2 Q13822 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
CYP19A1 P11511 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19003467 0.79 PORCN (0.54) MEN1ALOX15TSHRKMT2APORCN
SCHEMBL6660795 0.67 MEN1 (1.00) MEN1ALOX15TSHRKMT2APORCN
SCHEMBL27958208 0.67 CYP11B1 (0.54) MEN1ALOX15TSHRKMT2APORCN
Water SCHEMBL6337291 0.66 MEN1 (0.96) MEN1ALOX15TSHRKMT2APORCN
SCHEMBL28484940 0.65 CYP3A4 (0.71) MEN1ALOX15TSHRKMT2APORCN
SCHEMBL18746528 0.64 CYP3A4 (0.65) MEN1ALOX15TSHRKMT2ACYP3A4
SCHEMBL451 0.64 CYP3A4 (1.00) MEN1ALOX15TSHRKMT2ACYP3A4
SCHEMBL24782873 0.63 LMNA (0.55) MEN1ALOX15TSHRKMT2APORCN
SCHEMBL8392726 0.63 CYP3A4 (0.69) MEN1ALOX15TSHRKMT2ACYP3A4
SCHEMBL2604923 0.63 CYP3A4 (0.69) MEN1ALOX15TSHRKMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed