SCHEMBL190036

SCHEMBL190036

O=C(O)NC(c1ccccc1)C(O)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.48
MAPK1 P28482 1/20 0.48
KEAP1 Q14145 4/20 0.46
NFE2L2 Q16236 4/20 0.46
CYP2D6 P10635 1/20 0.45
SRC P12931 1/20 0.45
HPGD P15428 1/20 0.44
TP53 P04637 1/20 0.42
AOC3 Q16853 1/20 0.42
HDAC1 Q13547 2/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL162139 1.00 LMNA (0.48) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL14691171 1.00 LMNA (0.48) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL571797 1.00 LMNA (0.48) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL28707494 0.85 LMNA (0.52) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL12180786 0.85 LMNA (0.49) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL27486731 0.85 LMNA (0.49) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL7139715 0.85 SRC (0.47) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL8070685 0.85 SRC (0.47) LMNAMAPK1KEAP1NFE2L2CYP2D6
SCHEMBL8108955 0.83 LMNA (0.67) LMNAHPGDTP53HDAC1
SCHEMBL530337 0.83 LMNA (0.67) LMNAHPGDTP53HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 84 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2337561-A1 USE OF TOCOTRIENOL COMPOSITION FOR THE PREVENTION OF CANCER Davos Life Science Pte. Ltd. (SG) 2011-06-29 EP claimed
WO-2010047663-A1 USE OF TOCOTRIENOL COMPOSITION FOR THE PREVENTION OF CANCER DAVOS LIFE SCIENCE PTE. LTD. (SG) 2010-04-29 WO claimed
EP-4706770-A2 COMBINATION COMPRISING AN MEK INHIBITOR AND A B-RAF INHIBITOR Novartis AG (CH) 2026-03-11 EP disclosed
EP-4265300-B1 COMPOSITION COMPRISING A 17 A-HYDROXYLASE/C17,20 LYASE (CYP17A1) INHIBITOR AND AN AKT INHIBITOR NOVARTIS AG (CH) 2025-12-10 EP disclosed
WO-2025235719-A1 DIMERIC SMAC MIMETICS USEFUL IN HIV THERAPY VIIV HEALTHCARE COMPANY (US) 2025-11-13 WO disclosed
EP-4397376-A2 COMBINATION COMPRISING AN MEK INHIBITOR AND A B-RAF INHIBITOR Novartis AG (CH) 2024-07-10 EP disclosed
EP-3468953-B1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE IP DEV LTD (GB) 2024-05-22 EP disclosed
EP-4159217-B1 COMBINATION COMPRISING AN MEK INHIBITOR AND A B-RAF INHIBITOR NOVARTIS AG (CH) 2024-05-22 EP disclosed
EP-4342473-A2 COMPOUNDS USEFUL IN HIV THERAPY GlaxoSmithKline Intellectual Property Development Limited (GB) 2024-03-27 EP disclosed
EP-4159205-B1 NOVEL PHARMACEUTICAL COMPOSITION NOVARTIS AG (CH) 2024-02-14 EP disclosed
EP-4159204-B1 NOVEL PHARMACEUTICAL COMPOSITION NOVARTIS AG (CH) 2024-02-14 EP disclosed
US-7332617-B2 Process for the preparation of docetaxel trihydrate SHANGHAI DESANO CHEMICAL PHARMACEUTICAL CO., LTD. (CN) 2008-02-19 US disclosed
US-20070197538-A1 Anti-vascular and anti-proliferation methods, therapies, and combinations employing specific tyrosine kinase inhibitors AVENTIS PHARMA S.A. (FR) 2007-08-23 US disclosed
WO-2006128740-A2 ANTI-VASCULAR METHODS AND THERAPIES EMPLOYING LYSYL OXIDASE INHIBITORS CENTELION (FR) 2006-12-07 WO disclosed
US-20060217436-A1 Process for the preparation of docetaxel trihydrate SHANGHAI DESANO CHEMICAL PHARMACEUTICAL CO., LTD (CN) 2006-09-28 US disclosed
EP-1694660-A1 PROCESS FOR THE PREPARATION OF ANHYDROUS AND HYDRATED ACTIVE PHARMACEUTICAL INGREDIENTS (APIS); STABLE PHARMACEUTICAL COMPOSITIONS PREPARED FROM THE SAME AND USES OF SAID COMPOSITIONS Quiral Quimica Do Brasil (BR) 2006-08-30 EP disclosed
EP-1687642-A2 ANTI-VASCULAR AND ANTI-PROLIFERATION METHODS, THERAPIES, AND COMBINATIONS EMPLOYING SPECIFIC TYROSINE KINASE INHIBITORS CENTELION (FR) 2006-08-09 EP disclosed
EP-1623982-A1 THE PROCESS FOR THE PREPARATION OF DOCETAXEL TRIHYDRATE Shanghai Desano Chemical Pharmaceutical CO., Ltd. (CN) 2006-02-08 EP disclosed
WO-2005061474-A1 PROCESS FOR THE PREPARATION OF ANHYDROUS AND HYDRATED ACTIVE PHARMACEUTICAL INGREDIENTS (APIS); STABLE PHARMACEUTICAL COMPOSITIONS PREPARED FROM THE SAME AND USES OF SAID COMPOSITIONS QUIRAL QUÍMICA DO BRASIL (BR) 2005-07-07 WO disclosed
WO-2005038465-A2 ANTI-VASCULAR AND ANTI-PROLIFERATION METHODS, THERAPIES, AND COMBINATIONS EMPLOYING SPECIFIC TYROSINE KINASE INHIBITORS CENTELION (FR) 2005-04-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197538-A1 Anti-vascular and anti-proliferation methods, therapies, and combinations employing specific tyrosine kinase inhibitors MCL1, ABL1, TIE1 LMNA 2763/4885MAPK1 157/4885KEAP1 2868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.