SCHEMBL19003726

SCHEMBL19003726

CCCCC(CCCC)CN1CCN(c2ccc(F)cc2)C[C@H]1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
ALDH1A1 P00352 2/20 0.40
ADORA2A P29274 2/20 0.38
ADORA1 P30542 1/20 0.38
KCNH2 Q12809 1/20 0.38
GRM2 Q14416 1/20 0.38
DHFR P00374 2/20 0.37
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
GFER P55789 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NOTUM Q6P988 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897240 0.82 ADORA2A (0.41) ALDH1A1ADORA2AADORA1KCNH2SIGMAR1
SCHEMBL15857990 0.81 ESR1 (0.45) ALDH1A1ADORA2AADORA1KCNH2SIGMAR1
SCHEMBL15434161 0.74 KDM4E (0.42) ALDH1A1ADORA2AADORA1KCNH2SIGMAR1
SCHEMBL19003515 0.73 MAPT (0.39) ALDH1A1DHFRLMNAMAPTMAPK1
SCHEMBL15383525 0.70 ADRA2A (0.52) ALDH1A1LMNAMAPTMAPK1HTT
SCHEMBL27497948 0.70 ADRA2A (0.52) ALDH1A1LMNAMAPTMAPK1HTT
SCHEMBL15858027 0.70 ADRA2A (0.52) ALDH1A1LMNAMAPTMAPK1HTT
SCHEMBL17897235 0.69 MAPT (0.43) ALDH1A1LMNAMAPTMAPK1HTT
SCHEMBL15858970 0.69 MAPT (0.43) ALDH1A1LMNAMAPTMAPK1HTT
SCHEMBL18948442 0.69 ALDH1A1 (0.41) ALDH1A1LMNAMAPTMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2938344-B1 PIPERAZINE-SUBSTITUTED [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINE COMPOUNDS WITH A2A ANTAGONIST PROPERTIES MERCK SHARP & DOHME (US) 2017-06-21 EP disclosed