SCHEMBL19004877

SCHEMBL19004877

O=C(O)c1ccc2nc(Nc3cc(CN4CCNCC4)ccn3)[nH]c2c1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 20/20 0.62
IKBKE Q14164 3/20 0.62
CCNT1 O60563 1/20 0.57
CDK9 P50750 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19004878 0.90 TBK1 (0.62) TBK1IKBKECCNT1CDK9
Hydrochloric Acid SCHEMBL18985648 0.89 TBK1 (0.61) TBK1IKBKECCNT1CDK9
SCHEMBL18985814 0.86 TBK1 (0.79) TBK1
SCHEMBL19004994 0.84 TBK1 (0.66) TBK1IKBKE
SCHEMBL19005192 0.84 TBK1 (0.71) TBK1IKBKE
SCHEMBL18985932 0.84 TBK1 (0.80) TBK1IKBKE
Hydrochloric Acid SCHEMBL20720923 0.83 TBK1 (0.70) TBK1IKBKE
SCHEMBL19004876 0.83 NPSR1 (0.52) TBK1IKBKECCNT1CDK9
SCHEMBL19005014 0.82 POLB (0.51) TBK1IKBKECCNT1CDK9
SCHEMBL18985947 0.82 TBK1 (0.65) TBK1IKBKECCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed