SCHEMBL19004876

SCHEMBL19004876

O=C(O)c1ccc2nc(Nc3cc(CO)ccn3)[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.52
POLB P06746 1/20 0.49
TBK1 Q9UHD2 15/20 0.48
IKBKE Q14164 2/20 0.47
HSP90AA1 P07900 1/20 0.46
ESR2 Q92731 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
CCNT1 O60563 1/20 0.45
CDK9 P50750 1/20 0.45
AKR1C3 P42330 1/20 0.45
APEX1 P27695 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005014 0.90 POLB (0.51) NPSR1POLBTBK1IKBKEHSP90AA1
SCHEMBL18985777 0.88 KDM4E (0.48) TBK1IKBKE
SCHEMBL19004877 0.83 TBK1 (0.62) TBK1IKBKECCNT1CDK9
SCHEMBL4235671 0.81 ALDH1A1 (0.63) NPSR1POLBHSP90AA1ESR2TDP1
SCHEMBL18985935 0.81 TBK1 (0.59) TBK1IKBKECCNT1CDK9
Hydrochloric Acid SCHEMBL18985421 0.80 TBK1 (0.58) TBK1IKBKECCNT1CDK9
SCHEMBL18985814 0.79 TBK1 (0.79) TBK1
SCHEMBL18985710 0.78 TBK1 (0.47) TBK1IKBKE
SCHEMBL19004994 0.77 TBK1 (0.66) TBK1IKBKE
SCHEMBL4244217 0.77 AKR1C3 (0.52) NPSR1POLBHSP90AA1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed