SCHEMBL19005014

SCHEMBL19005014

O=C(O)c1ccc2nc(Nc3cc(CCl)ccn3)[nH]c2c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
TBK1 Q9UHD2 17/20 0.47
IKBKE Q14164 2/20 0.47
NPSR1 Q6W5P4 1/20 0.45
HSP90AA1 P07900 1/20 0.45
ESR2 Q92731 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CCNT1 O60563 1/20 0.45
CDK9 P50750 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19004876 0.90 NPSR1 (0.52) POLBTBK1IKBKENPSR1HSP90AA1
SCHEMBL18985710 0.88 TBK1 (0.47) TBK1IKBKE
SCHEMBL19004877 0.82 TBK1 (0.62) TBK1IKBKECCNT1CDK9
SCHEMBL19004879 0.81 TBK1 (0.45) TBK1IKBKECCNT1CDK9
SCHEMBL4235671 0.80 ALDH1A1 (0.63) POLBNPSR1HSP90AA1ESR2TDP1
SCHEMBL18985420 0.80 TBK1 (0.57) TBK1IKBKECCNT1CDK9
SCHEMBL18985777 0.78 KDM4E (0.48) TBK1IKBKE
SCHEMBL19004994 0.78 TBK1 (0.66) TBK1IKBKE
SCHEMBL18985814 0.78 TBK1 (0.79) TBK1
SCHEMBL4244217 0.76 AKR1C3 (0.52) POLBNPSR1HSP90AA1ESR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed