SCHEMBL19005522

SCHEMBL19005522

c1cc2c(nc3n2CCNC3)[nH]1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
HTR2C P28335 10/20 0.38
HTR2A P28223 9/20 0.38
MCHR1 Q99705 1/20 0.34
WNT1 P04628 1/20 0.31
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31
HTR6 P50406 1/20 0.31
CXCR4 P61073 1/20 0.30
AURKA O14965 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005520 0.73 HTR2A (0.35) HTR2CHTR2AMCHR1WNT1GSK3B
SCHEMBL19005518 0.73 HTR2A (0.35) HRH4HTR2CHTR2AMCHR1HTR6
SCHEMBL839815 0.71 HTR2A (0.50) HTR2CHTR2AMCHR1
SCHEMBL29539173 0.71 HTR2A (0.50) HTR2CHTR2AMCHR1
Hydrochloric Acid SCHEMBL20139551 0.70 HTR2A (0.49) HTR2CHTR2AMCHR1
SCHEMBL19005560 0.70 HTR2A (0.32) HRH4HTR2CHTR2AWNT1GSK3B
SCHEMBL31164710 0.70 HTR2A (0.56) HTR2CHTR2AMCHR1
SCHEMBL19005519 0.69 HTR2C (0.38) HTR2CHTR2AMCHR1
SCHEMBL19005525 0.69 HTR2C (0.37) HTR2CHTR2AMCHR1DYRK1A
SCHEMBL19005539 0.68 MCHR1 (0.37) HTR2CHTR2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101796-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed