SCHEMBL19005956

SCHEMBL19005956

CCCOc1cc2c(cc1C(=O)CCc1ccc(OC)c(N)c1)OCCS2(=O)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.36
SLC6A4 P31645 1/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC2 Q92769 2/20 0.36
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SLC5A1 P13866 1/20 0.34
SLC5A2 P31639 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP19A1 P11511 1/20 0.33
GAA P10253 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
CTNNB1 P35222 1/20 0.32
WNT3A P56704 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19005989 0.91 HDAC1 (0.37) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL18987192 0.87 CYP19A1 (0.44) HTR1ASLC6A4HDAC1HDAC2MEN1
SCHEMBL19005918 0.83 HTR1A (0.38) HTR1ASLC6A4MEN1KMT2ANPSR1
SCHEMBL19005957 0.82 HDAC1 (0.36) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL19005969 0.81 CYP19A1 (0.45) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL18987395 0.81 CHRM4 (0.37) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL18987197 0.80 HDAC1 (0.36) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL18987410 0.79 CYP3A4 (0.41) HDAC1HDAC2MEN1KMT2ANPSR1
SCHEMBL18987304 0.79 HDAC1 (0.39) HDAC1HDAC2MEN1KMT2ASLC5A1
SCHEMBL19005985 0.79 HDAC1 (0.39) HDAC1HDAC2MEN1KMT2ASLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103637-A1 DIPHENYLPROPANE COMPOUNDS AND THEIR CYTOTOXIC ACTIVITY BLIRT S.A. (PL) 2017-06-22 WO disclosed