SCHEMBL19013259

SCHEMBL19013259

CCc1cc(O)ccc1C1CCN(C(=O)C(C)O)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GUCY1A1 Q02108 4/20 0.41
GUCY1B1 Q02153 4/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40
SLC9A1 P19634 1/20 0.40
CCR1 P32246 2/20 0.38
MGLL Q99685 2/20 0.37
ROCK2 O75116 1/20 0.37
DRD2 P14416 2/20 0.36
ADAM17 P78536 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36
PDE4B Q07343 1/20 0.35
DRD3 P35462 1/20 0.35
NAMPT P43490 1/20 0.35
KIF11 P52732 1/20 0.35
QDPR P09417 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17395670 0.84 MGLL (0.40) CYP3A4CYP2C9SLC9A1MGLLDRD2
SCHEMBL20847810 0.83 HSD17B10 (0.53) CCR1ADAMTS5
SCHEMBL17397714 0.82 TDP1 (0.47) GUCY1A1GUCY1B1CYP3A4CYP2C9SLC9A1
SCHEMBL2480697 0.79 CYP3A4 (0.48) CYP3A4CYP2C9SLC9A1PDE4BNAMPT
SCHEMBL19013103 0.78 MAPT (0.50) CYP3A4CYP2C9
SCHEMBL17398252 0.75 MGLL (0.41) SLC9A1MGLLDRD2DRD3
SCHEMBL3143892 0.74 NUDT1 (0.40) DRD2DRD3
SCHEMBL19012974 0.74 ADAMTS5 (0.43) GUCY1A1GUCY1B1CYP3A4CYP2C9SLC9A1
SCHEMBL28134205 0.72 SLC6A2 (0.43) QDPR
SCHEMBL3809683 0.72 ESR2 (0.51) CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103888-A1 INDANE DERIVATIVES AND THE USE THEREOF AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS NOVARTIS AG (CH) 2017-06-22 WO disclosed