Odevixibat

Odevixibat

SCHEMBL19046540

CCCCC1(CCCC)CN(c2ccccc2)c2cc(SC)c(OCC(=O)NC(C(=O)N[C@@H](CC)C(=O)O)c3ccc(O)cc3)cc2S(=O)(=O)N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC10A2

The experimentally established mechanism targets of Odevixibat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC10A2 known ✓ Q12908 2/20 0.31
NR1H4 Q96RI1 1/20 1.00
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Odevixibat SCHEMBL946468 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL25794588 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL17733623 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL31121705 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL16414427 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
SCHEMBL20260213 0.99 NR1H4 (0.98) NR1H4KMT2AATMSLC10A2
SCHEMBL4566711 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL19046549 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL918882 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL2697206 0.96 NR1H4 (0.92) NR1H4KMT2AATMSLC10A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240207260-A1 METHODS FOR TREATING CHOLESTASIS MIRUM PHARMACEUTICALS, INC. (US) 2024-06-27 US disclosed
US-10221212-B2 IBAT inhibitors for the treatment of liver diseases ALBIREO AB (SE) 2019-03-05 US disclosed
US-20170182059-A1 IBAT Inhibitors for the Treatment of Liver Disease ALBIREO AB (SE) 2017-06-29 US disclosed
US-20170182115-A1 PHARMACEUTICAL COMBINATION COMPRISING AN IBAT INHIBITOR AND A BILE ACID BINDER ALBIREO AB (SE) 2017-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10221212-B2 IBAT inhibitors for the treatment of liver diseases GPR119, SLC10A1, SLC10A2 SLC10A2 3/4885NR1H4 46/4885KMT2A 1882/4885
US-20170182115-A1 PHARMACEUTICAL COMBINATION COMPRISING AN IBAT INHIBITOR AND A BILE ACID BINDER SLC10A2, GIPR, GPBAR1 SLC10A2 1/4885NR1H4 8/4885KMT2A 3354/4885
US-20170182059-A1 IBAT Inhibitors for the Treatment of Liver Disease SLC10A2, SLC10A1, GPR119 SLC10A2 1/4885NR1H4 50/4885KMT2A 1853/4885
US-20240207260-A1 METHODS FOR TREATING CHOLESTASIS SLC10A1, SLC10A2, NR1H4 SLC10A2 2/4885NR1H4 3/4885KMT2A 3031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.