Odevixibat

Odevixibat

SCHEMBL946468

CCCCC1(CCCC)CN(c2ccccc2)c2cc(SC)c(OCC(=O)N[C@@H](C(=O)N[C@@H](CC)C(=O)O)c3ccc(O)cc3)cc2S(=O)(=O)N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC10A2

The experimentally established mechanism targets of Odevixibat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC10A2 known ✓ Q12908 2/20 0.31
NR1H4 Q96RI1 1/20 1.00
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Odevixibat SCHEMBL19046540 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL25794588 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL17733623 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL31121705 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
Odevixibat SCHEMBL16414427 1.00 NR1H4 (1.00) NR1H4KMT2AATMSLC10A2
SCHEMBL20260213 0.99 NR1H4 (0.98) NR1H4KMT2AATMSLC10A2
SCHEMBL4566711 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL19046549 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL918882 0.96 NR1H4 (0.93) NR1H4SLC10A2
SCHEMBL2697206 0.96 NR1H4 (0.92) NR1H4KMT2AATMSLC10A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 846 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724071-A1 NOVEL USE OF AN ILEAL BILE ACID TRANSPORTER INHIBITOR FOR THE TREATMENT OF PRURITUS GlaxoSmithKline Intellectual Property (No. 2) Limited (GB) 2026-04-15 EP claimed
US-20260091040-A1 Treating Progressive Familial Intrahepatic Cholestasis (PFIC) with IBAT Inhibitors ALBIREO AB (SE) 2026-04-02 US claimed
US-12508234-B2 Pharmaceutical formulation of odevixibat ALBIREO AB (SE) 2025-12-30 US claimed
US-12447156-B2 Treating progressive familial intrahepatic cholestasis (PFIC) with IBAT inhibitors ALBIREO AB (SE) 2025-10-21 US claimed
EP-4629997-A1 ASBT INHIBITORS IN THE TREATMENT OF RENAL DISEASES Albireo AB (SE) 2025-10-15 EP claimed
EP-4630112-A1 COCRYSTALS OF ODEVIXIBAT Albireo AB (SE) 2025-10-15 EP claimed
EP-4590314-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS Astellas Gene Therapies, Inc. (US) 2025-07-30 EP claimed
EP-4566590-A1 TASTE-MASKING MICROSPHERE, PREPARATION PROCESS THEREFOR, AND USE THEREOF Harbin Kanon Pharmaceutical Co., Ltd (CN) 2025-06-11 EP claimed
EP-4511038-A1 SUBCUTANEOUS ADMINISTRATION OF AN ASBT INHIBITOR Albireo AB (SE) 2025-02-26 EP claimed
US-20250019354-A1 Crystal Modifications of Odevixibat ALBIREO AB (SE) 2025-01-16 US claimed
US-20050171204-A1 Substituted phenylpropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor alpha (ppar) ASTRAZENECA AB (SE) 2005-08-04 US claimed
US-20050131068-A1 Therapeutic agents ASTRAZENECA AB (SE) 2005-06-16 US claimed
EP-1539120-A1 COMBINATION OF AN IBAT INHIBITOR AND A METAL SALT FOR THE TREATMENT OF DIARRHOEA Astrazeneca AB (SE) 2005-06-15 EP claimed
US-20050113362-A1 Substituted phenypropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor alpha (ppar) ASTRAZENECA AB R & D HEADQUARTERS - GLOBAL IINTELLECTUAL PROPERT (SE) 2005-05-26 US claimed
WO-2004089350-A1 USE OF AN IBAT INHIBITOR FOR THE TREATMENT OF PROPHYLAXIS OF CONSTIPATION ASTRAZENECA AB (SE) 2004-10-21 WO claimed
EP-1458677-A1 3-PHENYL-2-ARYLALKYLTHIOPROPIONIC ACID DERIVATIVES AS SELECTIVE AGONISTS OF PPAR-ALPHA Astrazeneca AB (SE) 2004-09-22 EP claimed
EP-1458672-A1 SUBSTITUTED PHENYLPROPIONIC ACID DERIVATIVES AS AGONISTS TO HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA(PPAR) AstraZeneca AB (SE) 2004-09-22 EP claimed
WO-2004006899-A1 COMBINATION OF AN IBAT INHIBITOR AND A METAL SALT FOR THE TREATMENT OF DIARRHOEA ASTRAZENECA AB (SE) 2004-01-22 WO claimed
WO-2003051826-A1 3-PHENYL-2-ARYLALKYLTHIOPROPIONIC ACID DERIVATIVES AS SELECTIVE AGONISTS OF PPAR-ALPHA ASTRAZENECA AB (SE) 2003-06-26 WO claimed
WO-2003051822-A1 SUBSTITUTED PHENYLPROPIONIC ACID DERIVATIVES AS AGONISTS TO HUMAN PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR ALPHA (PPAR) ASTRAZENECA AB (SE) 2003-06-26 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050131068-A1 Therapeutic agents GPR119, INSR, LIPA SLC10A2 175/4885NR1H4 94/4885KMT2A 3639/4885
US-12508234-B2 Pharmaceutical formulation of odevixibat SLC10A1, ABCB11, SLC10A2 SLC10A2 3/4885NR1H4 39/4885KMT2A 3186/4885
US-12447156-B2 Treating progressive familial intrahepatic cholestasis (PFIC) with IBAT inhibitors SLC10A1, SLC10A2, ABCB11 SLC10A2 2/4885NR1H4 4/4885KMT2A 1279/4885
US-20050113362-A1 Substituted phenypropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor alpha (ppar) PPARA, PPARD, PPARG SLC10A2 434/4885NR1H4 33/4885KMT2A 2757/4885
US-20260091040-A1 Treating Progressive Familial Intrahepatic Cholestasis (PFIC) with IBAT Inhibitors SLC10A2, SLC10A1, ABCB11 SLC10A2 1/4885NR1H4 26/4885KMT2A 2489/4885
US-20050171204-A1 Substituted phenylpropionic acid derivatives as agonists to human peroxisome proliferator-activated receptor alpha (ppar) PPARA, PPARD, PPARG SLC10A2 209/4885NR1H4 46/4885KMT2A 3897/4885
US-20250019354-A1 Crystal Modifications of Odevixibat OR10J3, SULT1E1, OPRD1 SLC10A2 1148/4885NR1H4 841/4885KMT2A 496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.