SCHEMBL1905136

SCHEMBL1905136

CCC(C)C(NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1cccc2ccccc12)C(=O)NCc1cnc(N)s1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.53
CTSS P25774 1/20 0.53
CYP3A4 P08684 2/20 0.45
MME P08473 1/20 0.44
ACE P12821 1/20 0.44
CPA1 P15085 1/20 0.44
ACE2 Q9BYF1 1/20 0.44
REN P00797 13/20 0.43
CTSD P07339 1/20 0.42
PSMB1 P20618 1/20 0.42
PSMB8 P28062 1/20 0.42
PSMB9 P28065 1/20 0.42
PSMB5 P28074 1/20 0.42
PSMB10 P40306 1/20 0.42
PSMB2 P49721 1/20 0.42
CTSB P07858 1/20 0.41
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1905139 1.00 CTSK (0.53) CTSKCTSSCYP3A4MMEACE
SCHEMBL1905137 1.00 CTSK (0.53) CTSKCTSSCYP3A4MMEACE
SCHEMBL1908220 0.91 CTSS (0.64) CTSKCTSSCYP3A4PSMB1PSMB8
SCHEMBL1432298 0.87 CTSK (0.53) CTSKCTSSCYP3A4MMEACE
SCHEMBL1432294 0.87 CTSK (0.53) CTSKCTSSCYP3A4MMEACE
SCHEMBL1432297 0.87 CTSK (0.53) CTSKCTSSCYP3A4MMEACE
SCHEMBL1905660 0.85 MME (0.51) CTSKCTSSMMEACECPA1
SCHEMBL1907287 0.81 MME (0.51) CTSKCTSSMMEACECPA1
SCHEMBL1905678 0.80 MME (0.43) CTSKCTSSMMEACECPA1
SCHEMBL1432788 0.76 CTSS (0.65) CTSKCTSSCYP3A4PSMB1PSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051673-A1 AMINOTHIAZOLE DERIVATIVES USEFUL AS KLK1 INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed