SCHEMBL19059003

SCHEMBL19059003

CC1(C)CCc2cncnc2C1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.40
LIMK1 P53667 1/20 0.35
HDAC9 Q9UKV0 1/20 0.33
CNR2 P34972 1/20 0.33
CES1 P23141 1/20 0.32
PDK1 Q15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21983728 0.86 CYP11B2 (0.38) CYP11B2HDAC9
SCHEMBL9538975 0.85 HDAC9 (0.41) CYP11B2LIMK1HDAC9CES1PDK1
SCHEMBL19059299 0.82 CYP11B2 (0.36) CYP11B2HDAC9
SCHEMBL16461043 0.79 HDAC9 (0.32) CYP11B2HDAC9
SCHEMBL19059295 0.79 CYP11B2 (0.36) CYP11B2HDAC9
SCHEMBL19059004 0.77 HDAC9 (0.36) CYP11B2HDAC9
SCHEMBL15492413 0.75 CYP11B2 (0.36) CYP11B2HDAC9
SCHEMBL15492457 0.74 CYP11B2 (0.36) CYP11B2HDAC9
SCHEMBL9770510 0.73 DRD2 (0.33) LIMK1CNR2CES1PDK1
SCHEMBL16984843 0.73 CYP11B2 (0.33) CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2693882-B1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK SHARP & DOHME (US) 2017-06-28 EP disclosed