SCHEMBL1906017

SCHEMBL1906017

Cc1ccccc1OCC(=O)N[C@@H](Cc1cccc2ccccc12)C(=O)NCc1ccc(N)nc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.46
POLB P06746 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK1 P28482 1/20 0.43
TP53 P04637 1/20 0.43
OPRD1 P41143 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
TACR1 P25103 1/20 0.41
LCK P06239 2/20 0.40
PSMB8 P28062 1/20 0.40
PSMB5 P28074 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1901459 0.89 OPRD1 (0.45) SMN1; SMN2OPRD1CTSSCTSKTACR1
SCHEMBL1905963 0.86 LCK (0.48) MAPTKMT2AMAPK1OPRD1KDM4E
SCHEMBL1905965 0.86 LCK (0.48) MAPTKMT2AMAPK1OPRD1KDM4E
SCHEMBL1906797 0.86 OPRD1 (0.47) OPRD1CTSSCTSKTACR1LCK
SCHEMBL1906792 0.86 OPRD1 (0.47) OPRD1CTSSCTSKTACR1LCK
SCHEMBL1904790 0.84 OPRD1 (0.48) OPRD1CTSSCTSKLCKPSMB8
SCHEMBL1904838 0.83 TACR1 (0.44) MEN1MAPTKMT2ATP53OPRD1
SCHEMBL1902805 0.82 OPRD1 (0.46) OPRD1CTSSCTSKLCKPSMB8
SCHEMBL1902802 0.82 OPRD1 (0.46) OPRD1CTSSCTSKLCKPSMB8
SCHEMBL1905132 0.81 PSMB8 (0.53) OPRD1CTSSCTSKLCKPSMB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO claimed
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed