SCHEMBL19063

SCHEMBL19063

FC(F)(F)c1nccc(Cl)n1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 8/20 0.46
IDH1 O75874 5/20 0.38
IDH2 P48735 4/20 0.38
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757680 1.00 MALT1 (0.46) MALT1IDH1IDH2CYP3A4CYP2C9
SCHEMBL2649999 0.83 MALT1 (0.33) MALT1IDH1IDH2
SCHEMBL30755800 0.83 MAP4K1 (0.35) MALT1IDH1IDH2
SCHEMBL11113890 0.77 ADORA2A (0.34) CYP3A4
SCHEMBL21328933 0.74 MALT1 (0.52) MALT1IDH1IDH2NOS3NOS2
SCHEMBL3295825 0.74 MALT1 (0.47) MALT1IDH1IDH2TAS2R14
SCHEMBL31493074 0.74 TAAR1 (0.32) CYP3A4CYP2C19
SCHEMBL19337822 0.73 MALT1 (0.46) MALT1IDH1IDH2NOS3NOS2
SCHEMBL1420222 0.73 NOS3 (0.47) MALT1IDH1IDH2KCNH2NOS3
SCHEMBL18428 0.73 MALT1 (0.46) MALT1IDH1IDH2NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 577 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102911123-B Preparation method of 2-chloro trifluoromethyl pyrimidine compound SHANGHAI TITAN TECHNOLOGY CO LTD 2015-04-22 CN claimed
CN-102911123-A Preparation method of 2-chloro trifluoromethyl pyrimidine compound SHANGHAI TITAN TECHNOLOGY CO LTD 2013-02-06 CN claimed
CN-1057651-A The preparation method of pyrimidine compound BRISTOL MYERS SQUIBB CO (US) 1992-01-08 CN claimed
EP-0463596-A1 Cerebral function enhancing pyrimidinyl derivatives Bristol-Myers Squibb Company (US) 1992-01-02 EP claimed
US-20260083851-A1 POTENT ASGPR-BINDING HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF IMMUNOGLOBULINS AND OTHER PROTEINS AVILAR THERAPEUTICS, INC. (US) 2026-03-26 US disclosed
US-20260042749-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2026-02-12 US disclosed
US-12545659-B2 IRAK degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2026-02-10 US disclosed
US-12539295-B2 IRAK degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2026-02-03 US disclosed
US-20250333417-A1 IRAK DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2025-10-30 US disclosed
US-12433895-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2025-10-07 US disclosed
US-12390463-B2 Dosage forms and regimens for amino acid compounds PLIANT THERAPEUTICS, INC. (US) 2025-08-19 US disclosed
EP-4598923-A1 SUPRAMOLECULAR POLYMER THERAPEUTICS AND DIAGNOSTICS The Regents of the University of California (US) 2025-08-13 EP disclosed
US-4137237-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-01-30 US disclosed
US-4137234-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-01-30 US disclosed
US-4070475-A THIOALKYL-, AMINOALKYL-, AND OXYALKYL- SUBSTITUTED GUANIDINES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1978-01-24 US disclosed
US-4024271-A INHIBITORS OF HISTAMINE ACTIVITY SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-05-17 US disclosed
US-4022797-A PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-05-10 US disclosed
US-4018931-A INHIBITION OF H-2 HISTAMINE RECEPTORS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-04-19 US disclosed
US-3950353-A HISTAMINE INHIBITORS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-04-13 US disclosed
US-3950333-A HISTAMINE INHIBITORS, OXYALKYL, THIOALKYL, AMINOALKYL DERIVATIVES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12545659-B2 IRAK degraders and uses thereof IRAK2, IRAK3, IRAK4 MALT1 976/4885IDH1 1750/4885IDH2 1858/4885
US-12433895-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT MALT1 822/4885IDH1 172/4885IDH2 110/4885
US-12390463-B2 Dosage forms and regimens for amino acid compounds ITGB6, ITGA6, ITGAV MALT1 4670/4885IDH1 2011/4885IDH2 3408/4885
US-12539295-B2 IRAK degraders and uses thereof IRAK2, IRAK4, IRAK3 MALT1 339/4885IDH1 1526/4885IDH2 1437/4885
US-20260083851-A1 POTENT ASGPR-BINDING HETEROBIFUNCTIONAL COMPOUNDS FOR THE DEGRADATION OF IMMUNOGLOBULINS AND OTHER PROTEINS ASGR1, FCGR2A, FCGR3B MALT1 949/4885IDH1 3530/4885IDH2 4451/4885
US-20260042749-A1 IRAK DEGRADERS AND USES THEREOF IRAK2, IRAK3, IRAK4 MALT1 958/4885IDH1 1508/4885IDH2 1305/4885
US-20250333417-A1 IRAK DEGRADERS AND USES THEREOF IRAK2, IRAK3, IRAK1 MALT1 1097/4885IDH1 2500/4885IDH2 2900/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.