Elinafide

Elinafide

SCHEMBL19067

O=C1c2cccc3cccc(c23)C(=O)N1CCNCCCNCCN1C(=O)c2cccc3cccc(c23)C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 3/20 1.00
HEXA P06865 14/20 0.90
HEXB P07686 14/20 0.90
OGA O60502 1/20 0.90
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
NR1I2 O75469 1/20 0.57
POLB P06746 1/20 0.57
AHR P35869 1/20 0.57
RAD52 P43351 1/20 0.57
RCE1 Q9Y256 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Elinafide SCHEMBL6256967 1.00 SIRT1 (1.00) SIRT1HEXAHEXBOGAMEN1
Elinafide SCHEMBL29441732 1.00 SIRT1 (1.00) SIRT1HEXAHEXBOGAMEN1
SCHEMBL8396162 0.97 SIRT1 (0.94) SIRT1HEXAHEXBOGAMEN1
SCHEMBL31011151 0.95 HEXA (1.00) SIRT1HEXAHEXBOGA
SCHEMBL4408773 0.95 HEXA (1.00) SIRT1HEXAHEXBOGA
Bnipdpta SCHEMBL13909966 0.94 SIRT1 (0.88) SIRT1HEXAHEXBOGAMEN1
SCHEMBL13909979 0.94 SIRT1 (0.88) SIRT1HEXAHEXBOGAMEN1
SCHEMBL3290712 0.93 SIRT1 (0.86) SIRT1HEXAHEXBOGA
SCHEMBL14524900 0.93 SIRT1 (0.86) SIRT1HEXAHEXBOGANR1I2
Bnipspd SCHEMBL13909975 0.92 SIRT1 (0.91) SIRT1HEXAHEXBOGAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3065 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260083866-A1 COMPOSITIONS TARGETING ENDOTHELIAL CELLS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2026-03-26 US claimed
US-20260055182-A1 ANTI-L1-CAM ANTIBODIES AND THEIR USES FOR DIAGNOSTIC AND THERAPEUTIC APPLICATIONS CIS BIOPHARMA AG (CH) 2026-02-26 US claimed
US-20250326856-A1 HUMANIZED ANTI-CD45 ANTIBODIES AND USES THEREOF Fred Hutchison Cancer Center (US) 2025-10-23 US claimed
EP-4615580-A1 ANTI-L1-CAM ANTIBODIES AND THEIR USES FOR DIAGNOSTIC AND THERAPEUTIC APPLICATIONS CIS Biopharma AG (CH) 2025-09-17 EP claimed
US-12398402-B2 Reducing CD33 expression to selectively protect therapeutic cells FRED HUTCHINSON CANCER CENTER (US) 2025-08-26 US claimed
US-20250249125-A1 ANTI-CD90 ANTIBODIES, BINDING FRAGMENTS, AND USES THEREOF Fred Hutchison Cancer Center (US) 2025-08-07 US claimed
WO-2025097015-A1 CLEC2A-BINDING THERAPEUTICS FRED HUTCHINSON CANCER CENTER (US) 2025-05-08 WO claimed
WO-2025080875-A1 CYTOMEGALOVIRUS-DERIVED CD44 BINDING PROTEINS AND USES THEREOF LIONS EYE INSTITUTE (AU) 2025-04-17 WO claimed
WO-2025076048-A1 ANTI-CD90 ANTIBODIES, BINDING FRAGMENTS, AND USES THEREOF FRED HUTCHINSON CANCER CENTER (US) 2025-04-10 WO claimed
WO-2025036876-A2 NEW ANTI-CANCER APPROACHES ONA Therapeutics S.L. (ES) 2025-02-20 WO claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20060035945-A1 Triheterocyclic compounds, compositions, and methods for treating cancer or viral diseases INVESTISSEMENT QUEBEC (CA) 2006-02-16 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
EP-1085891-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE Advanced Medicine, Inc. (US) 2001-03-28 EP claimed
WO-1999064054-A9 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE INC (US) 2000-03-02 WO claimed
WO-1999064054-A1 MULTIBINDING INHIBITORS OF TOPOISOMERASE ADVANCED MEDICINE, INC. (US) 1999-12-16 WO claimed