SCHEMBL1908125

SCHEMBL1908125

O=C(c1ccc(Nc2ccccc2)cc1)c1ccccc1O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 5/20 0.67
MAPK12 P53778 5/20 0.67
MAPK11 Q15759 5/20 0.67
MAPK14 Q16539 5/20 0.67
LIG1 P18858 1/20 0.65
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
KDM4E B2RXH2 2/20 0.53
HPGD P15428 2/20 0.53
HSD17B10 Q99714 2/20 0.53
LMNA P02545 2/20 0.53
TP53 P04637 1/20 0.53
HTT P42858 1/20 0.53
POLB P06746 2/20 0.51
STS P08842 1/20 0.51
CASP3 P42574 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
ALDH1A1 P00352 2/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1908387 0.91 LIG1 (0.79) MAPK13MAPK12MAPK11MAPK14LIG1
SCHEMBL6651304 0.88 LIG1 (0.59) MAPK13MAPK12MAPK11MAPK14LIG1
SCHEMBL1905196 0.86 LIG1 (0.61) MAPK13MAPK12MAPK11MAPK14LIG1
SCHEMBL29499085 0.84 LIG1 (0.87) LIG1MEN1KMT2AKDM4EHPGD
SCHEMBL21802003 0.84 LIG1 (0.87) LIG1MEN1KMT2AKDM4EHPGD
SCHEMBL1906899 0.84 NPC1 (0.61) LIG1MEN1KMT2AKDM4EHPGD
SCHEMBL6653266 0.83 HPGD (0.57) LIG1MEN1KMT2AHPGDPOLB
SCHEMBL27555322 0.83 MAPK13 (0.62) MAPK13MAPK12MAPK11MAPK14MEN1
SCHEMBL28027482 0.83 LIG1 (0.77) LIG1MEN1KMT2AKDM4EHPGD
SCHEMBL22129808 0.82 LIG1 (0.76) LIG1MEN1KMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4684515-B2 2011-05-18 JP claimed
EP-1237845-B1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1BETA AND TNF-ALPHA LEO PHARMA AS (DK) 2007-05-23 EP claimed
US-20030013770-A1 Aminobenzophenones as inhibitors of il 1b and tnf LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 2003-01-16 US claimed
EP-1237845-A1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1BETA AND TNF-ALPHA LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2002-09-11 EP claimed
WO-2001042189-A1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1β AND TNF-$g(a) LEO PHARMA A/S (DK) 2001-06-14 WO claimed
EP-1237845-B1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1BETA AND TNF-ALPHA LEO PHARMA AS (DK) 2007-05-23 EP disclosed
US-6541670-B2 Antiinflammatory agents LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 2003-04-01 US disclosed
US-20030013770-A1 Aminobenzophenones as inhibitors of il 1b and tnf LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 2003-01-16 US disclosed
EP-1237845-A1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1BETA AND TNF-ALPHA LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2002-09-11 EP disclosed
WO-2001042189-A1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1β AND TNF-$g(a) LEO PHARMA A/S (DK) 2001-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030013770-A1 Aminobenzophenones as inhibitors of il 1b and tnf IL1B, IL1A, IL6 MAPK13 2221/4885MAPK12 1892/4885MAPK11 1835/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.