SCHEMBL19085282

SCHEMBL19085282

COCC1COc2ccc(C3(C(=O)OC)CC3)cc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.38
CYP3A4 P08684 4/20 0.36
MAP3K14 Q99558 2/20 0.36
CYP19A1 P11511 4/20 0.34
MAPT P10636 3/20 0.34
HPGD P15428 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ALOX15 P16050 2/20 0.34
ALOX12 P18054 2/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HRH3 Q9Y5N1 1/20 0.31
HDAC1 Q13547 1/20 0.31
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19753195 0.87 MAOB (0.37) MAOBCYP3A4MAP3K14CYP19A1MAPT
SCHEMBL29654008 0.78 MAOB (0.41) MAOBCYP3A4CYP19A1MAPTHPGD
SCHEMBL22997336 0.78 MAOB (0.41) MAOBCYP3A4CYP19A1MAPTHPGD
SCHEMBL19085860 0.76 MTNR1A (0.47) MAPTTP53
SCHEMBL1464653 0.76 MAOB (0.40) MAOBHPGDALDH1A1SMN1; SMN2
SCHEMBL18764225 0.70 ACHE (0.33) HRH3
SCHEMBL19085245 0.70 CFTR (0.38)
SCHEMBL14458379 0.70 CFTR (0.53) MEN1KMT2AALDH1A1SMN1; SMN2HDAC1
SCHEMBL26133742 0.69 PPIA (0.45) MAOBCYP3A4MAPTMEN1KMT2A
SCHEMBL1465911 0.68 CFTR (0.43) SMN1; SMN2HDAC1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11639347-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-05-02 US disclosed
US-20230127655-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-04-27 US disclosed
US-10975061-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-04-13 US disclosed
US-20200115366-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED 2020-04-16 US disclosed
US-10239867-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-03-26 US disclosed
US-20180162842-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED 2018-06-14 US disclosed
US-9974781-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2018-05-22 US disclosed
US-9758510-B2 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-09-12 US disclosed
US-20170189389-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10975061-B2 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-11639347-B2 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-20170189389-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-20200115366-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-20180162842-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-20230127655-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885
US-10239867-B2 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 MAOB 3306/4885CYP3A4 1368/4885MAP3K14 4715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.