SCHEMBL19086034

SCHEMBL19086034

Cc1ccc(F)cc1CNC(O)c1cc2c(s1)CCNC2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNMT P11086 5/20 0.40
ITGB3 P05106 4/20 0.32
ITGA2B P08514 4/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
TPSAB1 Q15661 1/20 0.31
TPSD1 Q9BZJ3 1/20 0.31
TPSG1 Q9NRR2 1/20 0.31
CCNT1 O60563 1/20 0.30
CDK9 P50750 1/20 0.30
MELK Q14680 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086033 0.77 ALDH1A1 (0.51) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL20778382 0.66 PNMT (0.61) PNMTITGB3ITGA2BPARP1PARP2
SCHEMBL21236155 0.62 PNMT (0.63) PNMTPARP1PARP2TPSAB1TPSD1
SCHEMBL30199323 0.61 CD274 (0.51) PNMTMELK
SCHEMBL29097942 0.61 CD274 (0.51) PNMTMELK
SCHEMBL6424327 0.61 PNMT (1.00) PNMTTPSAB1TPSD1TPSG1
SCHEMBL14035157 0.59 SLC6A4 (0.59)
SCHEMBL698730 0.58 SHBG (0.41)
SCHEMBL12538638 0.58 PNMT (0.49) PNMTITGB3ITGA2B
SCHEMBL17545266 0.58 PNMT (0.61) PNMTITGB3ITGA2BPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed