SCHEMBL19086245

SCHEMBL19086245

CNC(=O)c1cc2c(s1)CCN(C(=O)CNC(=O)c1ccc(N)c(C=N)c1)C2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.43
KDM1A O60341 5/20 0.43
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PRMT5 O14744 7/20 0.39
WDR77 Q9BQA1 7/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
F2 P00734 1/20 0.38
TPSAB1 Q15661 1/20 0.38
TPSD1 Q9BZJ3 1/20 0.38
TPSG1 Q9NRR2 1/20 0.38
THRB P10828 1/20 0.38
VDR P11473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19087005 0.91 KDM1A (0.41) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086019 0.89 ALDH1A1 (0.41) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086204 0.89 ALDH1A1 (0.43) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086203 0.88 PRMT5 (0.40) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086189 0.86 PRMT5 (0.48) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086218 0.85 KDM1A (0.48) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086195 0.85 KDM1A (0.41) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086253 0.85 KDM1A (0.41) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086202 0.84 KDM1A (0.48) HDAC6KDM1AALDH1A1L3MBTL1HTT
SCHEMBL19086315 0.84 KDM1A (0.47) HDAC6KDM1AALDH1A1L3MBTL1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed