SCHEMBL19086253

SCHEMBL19086253

N=Cc1cc(C(=O)NCC(=O)N2CCc3sc(C(=O)NC4CCNCC4)cc3C2)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.41
HDAC6 Q9UBN7 7/20 0.41
PRMT5 O14744 6/20 0.37
WDR77 Q9BQA1 6/20 0.37
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
NPC1 O15118 1/20 0.35
PRNP P04156 1/20 0.35
RAB9A P51151 1/20 0.35
F2 P00734 1/20 0.34
TPSAB1 Q15661 1/20 0.34
TPSD1 Q9BZJ3 1/20 0.34
TPSG1 Q9NRR2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086195 0.91 KDM1A (0.41) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086222 0.86 KDM1A (0.39) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086245 0.85 HDAC6 (0.43) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19087005 0.84 KDM1A (0.41) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086203 0.83 PRMT5 (0.40) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086189 0.82 PRMT5 (0.48) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086019 0.82 ALDH1A1 (0.41) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086204 0.82 ALDH1A1 (0.43) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086353 0.80 HDAC6 (0.43) KDM1AHDAC6PRMT5WDR77ALDH1A1
SCHEMBL19086216 0.80 HDAC6 (0.35) KDM1AHDAC6PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed