SCHEMBL19086255

SCHEMBL19086255

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)Nc3ccnc(C)c3)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ROCK2 O75116 4/20 0.38
MAOB P27338 6/20 0.38
LRRK2 Q5S007 2/20 0.37
ROCK1 Q13464 1/20 0.37
TRPV1 Q8NER1 2/20 0.37
MAOA P21397 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086178 0.93 NPC1 (0.38) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL19085999 0.90 TRPV1 (0.41) KMT2ANPC1RAB9AROCK2MAOB
SCHEMBL19085981 0.90 TRPV1 (0.41) KMT2ANPC1RAB9AROCK2MAOB
SCHEMBL19086349 0.90 MAOB (0.40) ROCK2MAOBROCK1
SCHEMBL19086167 0.89 METTL3 (0.37) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL19085977 0.89 NPC1 (0.45) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL19085989 0.88 MAOB (0.41) NPC1RAB9AROCK2MAOBROCK1
SCHEMBL19086169 0.88 METTL3 (0.37) MEN1KMT2ANPC1RAB9AL3MBTL1
SCHEMBL19085978 0.88 ROCK2 (0.46) NPC1RAB9AROCK2MAOBROCK1
SCHEMBL19086258 0.88 ROCK2 (0.34) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed