SCHEMBL19085989

SCHEMBL19085989

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)Nc3cccc(Cl)c3)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.41
ROCK2 O75116 4/20 0.40
ROCK1 Q13464 2/20 0.40
MAOA P21397 2/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CLK2 P49760 1/20 0.40
DYRK1A Q13627 1/20 0.40
PRKG1 Q13976 1/20 0.40
PRKD2 Q9BZL6 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
SGK2 Q9HBY8 1/20 0.40
STK17A Q9UEE5 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085999 0.92 TRPV1 (0.41) MAOBROCK2ROCK1MAOACLK2
SCHEMBL19085981 0.92 TRPV1 (0.41) MAOBROCK2ROCK1MAOACLK2
SCHEMBL19085978 0.92 ROCK2 (0.46) MAOBROCK2ROCK1MAOAMAP4K4
SCHEMBL19086255 0.88 MEN1 (0.39) MAOBROCK2ROCK1MAOANPC1
SCHEMBL19085977 0.88 NPC1 (0.45) MAOBROCK2ROCK1MAP4K4RPS6KB1
SCHEMBL19086178 0.87 NPC1 (0.38) MAOBROCK2ROCK1MAOAMAP4K4
SCHEMBL19086167 0.87 METTL3 (0.37) MAOBROCK2MAOANPC1RAB9A
SCHEMBL19086252 0.86 ROCK2 (0.37) MAOBROCK2ROCK1MAOAPRKD3
SCHEMBL19086169 0.86 METTL3 (0.37) MAOBROCK2ROCK1MAOANPC1
SCHEMBL19085993 0.86 BTK (0.38) ROCK2ROCK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed