SCHEMBL19086353

SCHEMBL19086353

N=C(F)c1cc(C(=O)NCC(=O)N2CCc3sc(C(=O)NC4CCCC4)cc3C2)ccc1N

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 8/20 0.43
KDM1A O60341 6/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PRNP P04156 1/20 0.37
F2 P00734 1/20 0.37
TPSAB1 Q15661 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PRMT5 O14744 4/20 0.36
WDR77 Q9BQA1 4/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086352 0.84 HDAC6 (0.40) HDAC6KDM1ANPC1RAB9ASMN1; SMN2
SCHEMBL19086195 0.80 KDM1A (0.41) HDAC6KDM1ANPC1RAB9AHTT
SCHEMBL19086253 0.80 KDM1A (0.41) HDAC6KDM1ANPC1RAB9AHTT
SCHEMBL19086222 0.79 KDM1A (0.39) HDAC6KDM1ANPC1RAB9AHTT
SCHEMBL19086995 0.77 ROCK2 (0.47) HDAC6KDM1ANPC1RAB9AHTT
SCHEMBL19086245 0.74 HDAC6 (0.43) HDAC6KDM1AHTTSMN1; SMN2F2
SCHEMBL19087005 0.73 KDM1A (0.41) HDAC6KDM1AHTTSMN1; SMN2ALDH1A1
SCHEMBL19086203 0.72 PRMT5 (0.40) HDAC6KDM1AHTTSMN1; SMN2ALDH1A1
SCHEMBL19086190 0.72 ROCK2 (0.48) HDAC6KDM1A
SCHEMBL19086189 0.71 PRMT5 (0.48) HDAC6KDM1AHTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed