SCHEMBL19087010

SCHEMBL19087010

N=Cc1cc(C(=O)NCC(=O)N2CCc3sc(C(=O)NCc4cccc5ccccc45)cc3C2)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.41
PRMT5 O14744 12/20 0.40
WDR77 Q9BQA1 12/20 0.40
CA2 P00918 1/20 0.38
HDAC6 Q9UBN7 3/20 0.38
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086315 0.89 KDM1A (0.47) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086245 0.83 HDAC6 (0.43) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086189 0.83 PRMT5 (0.48) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19087005 0.82 KDM1A (0.41) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086203 0.81 PRMT5 (0.40) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086202 0.80 KDM1A (0.48) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086204 0.80 ALDH1A1 (0.43) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086019 0.80 ALDH1A1 (0.41) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086238 0.80 EPHX2 (0.42) KDM1APRMT5WDR77HDAC6ALDH1A1
SCHEMBL19086218 0.80 KDM1A (0.48) KDM1APRMT5WDR77HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed