SCHEMBL19088009

SCHEMBL19088009

Oc1ccc2c(c1)NC(O)CC2

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 5/20 0.47
ESR1 P03372 3/20 0.47
DRD2 P14416 4/20 0.44
DRD3 P35462 3/20 0.44
OPRK1 P41145 2/20 0.44
DRD4 P21917 3/20 0.41
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726820 0.79 ESR2 (0.46) ESR2ESR1DRD2DRD3OPRK1
SCHEMBL13091390 0.79 DRD2 (0.39) ESR2ESR1DRD2
SCHEMBL2697405 0.76 MTNR1A (0.45)
SCHEMBL13305784 0.76 MTNR1A (0.45)
SCHEMBL21465771 0.75 GAA (0.44) ESR2ESR1DRD2DRD3OPRK1
Methane SCHEMBL10697109 0.74 MTNR1A (0.44)
SCHEMBL14409327 0.72 ESR2 (0.50) ESR2ESR1DRD2DRD3OPRK1
SCHEMBL5234926 0.72 ESR2 (0.50) ESR2ESR1DRD2DRD3OPRK1
SCHEMBL5235986 0.72 ESR2 (0.50) ESR2ESR1DRD2DRD3OPRK1
SCHEMBL5235983 0.72 ESR2 (0.50) ESR2ESR1DRD2DRD3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3397636-B1 PROCESS FOR THE PREPARATION OF QUINOLINE-2(1H)-ONE DERIVATIVES HONOUR R&D (IN) 2021-08-04 EP disclosed
WO-2017115287-A1 PROCESS FOR THE PREPARATION OF QUINOLINE-2(1H)-ONE DERIVATIVES HONOUR (R&D) (IN) 2017-07-06 WO disclosed