SCHEMBL19099129

SCHEMBL19099129

O=C(Cc1ccccc1F)N1CCc2cc(Br)cc([N+](=O)[O-])c21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.45
RAB9A P51151 2/20 0.45
MAPK1 P28482 3/20 0.42
MAPT P10636 5/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HTT P42858 1/20 0.39
EIF2AK3 Q9NZJ5 1/20 0.38
POLB P06746 1/20 0.38
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19099135 0.83 MAPK1 (0.45) L3MBTL1MAPK1MAPTSMN1; SMN2EIF2AK3
SCHEMBL30340615 0.79 ALDH1A1 (0.56) HTR2AHTR2CL3MBTL1MAPTSMN1; SMN2
SCHEMBL13041061 0.75 HTR2A (0.56) HTR2AHTR2CL3MBTL1RAB9AMAPK1
SCHEMBL3071409 0.75 HTR2A (0.56) HTR2AHTR2CL3MBTL1MAPTALDH1A1
SCHEMBL8909599 0.74 HTR2A (0.52) HTR2AHTR2CL3MBTL1MAPTSMN1; SMN2
SCHEMBL12919994 0.74 HTR2A (0.53) HTR2AHTR2CL3MBTL1MAPK1MAPT
SCHEMBL8905312 0.73 HTR2A (0.53) HTR2AHTR2CL3MBTL1MAPK1MAPT
SCHEMBL20865829 0.71 MAPK1 (0.64) MAPK1
SCHEMBL8905316 0.70 HTR2A (0.49) HTR2AHTR2CL3MBTL1MAPK1MAPT
SCHEMBL20897096 0.69 HTR2A (0.45) HTR2AHTR2CRAB9AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922405-B Compound with ERK kinase inhibitory activity, preparation method and application thereof 中国科学院上海药物研究所 2021-02-19 CN disclosed
WO-2017114510-A1 COMPOUND HAVING ERK KINASE INHIBITORY ACTIVITY, METHOD FOR PREPARATION THEREOF, AND USE THEREOF 中国科学院上海药物研究所 2017-07-06 WO disclosed