SCHEMBL19100596

SCHEMBL19100596

COC(=O)c1cc(-c2ccc(F)cc2)cn1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
IKBKB O14920 1/20 0.42
MAPT P10636 4/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CASP3 P42574 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19064181 0.82 KDR (0.44) KDM4EALDH1A1HSD17B10GAAALOX15
SCHEMBL20141700 0.71 KDM4E (0.36) KDM4EALDH1A1HSD17B10GAAMAPT
SCHEMBL12582220 0.71 NR4A2 (0.46) KDM4EALDH1A1GAAMAPTRAB9A
SCHEMBL19063822 0.70 LDHA (0.42) KDM4EALDH1A1HSD17B10ALOX15MAPT
SCHEMBL2952068 0.70 MEN1 (0.68) KDM4EALDH1A1SLC6A4SLC6A3MAPT
SCHEMBL4486670 0.69 KDM4E (0.57) KDM4EALDH1A1GAASLC6A4SLC6A3
SCHEMBL184208 0.69 KDM4E (0.61) KDM4EALDH1A1GAASLC6A4SLC6A3
SCHEMBL1254366 0.69 NR4A2 (0.54) KDM4EALDH1A1HSD17B10GAAALOX15
SCHEMBL28835928 0.68 SLC6A4 (0.50) KDM4ESLC6A4SLC6A3IKBKBMAPT
SCHEMBL19064093 0.68 KDR (0.44) KDM4EALDH1A1HSD17B10MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3400228-A1 FUSED QUADRACYCLIC COMPOUNDS, COMPOSITIONS AND USES THEREOF Tabomedex Biosciences, LLC (US) 2018-11-14 EP disclosed
WO-2017120164-A1 FUSED QUADRACYCLIC COMPOUNDS, COMPOSITIONS AND USES THEREOF Tabomedex Biosciences, LLC (US) 2017-07-13 WO disclosed