SCHEMBL20141700

SCHEMBL20141700

COC(=O)c1cc(Br)cn1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.36
NOTUM Q6P988 1/20 0.36
TSHR P16473 3/20 0.34
ALDH1A1 P00352 4/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
GAA P10253 3/20 0.34
NPSR1 Q6W5P4 2/20 0.34
POLB P06746 1/20 0.34
NR4A2 P43354 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
MAPK10 P53779 1/20 0.33
MAPK1 P28482 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30211465 0.80 L3MBTL1 (0.34) KDM4ENOTUMTSHRALDH1A1L3MBTL1
SCHEMBL4131647 0.79 NR1H2 (0.42) KDM4ENOTUML3MBTL1
SCHEMBL1254373 0.78 CYP1A2 (0.46) KDM4ENOTUMTSHRL3MBTL1NPSR1
SCHEMBL21587971 0.77 NOTUM (0.33) KDM4ENOTUMALDH1A1L3MBTL1GAA
SCHEMBL1966318 0.76 NPSR1 (0.37) KDM4ENOTUMTSHRALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL29155899 0.75 NPSR1 (0.36) KDM4ENOTUMTSHRALDH1A1L3MBTL1
SCHEMBL1003620 0.75 ALDH1A1 (0.41) KDM4EALDH1A1L3MBTL1GAANPSR1
SCHEMBL20562638 0.74 NR4A2 (0.42) KDM4ENOTUMTSHRALDH1A1NR4A2
SCHEMBL16142787 0.73 NR4A2 (0.49) KDM4ETSHRALDH1A1L3MBTL1GAA
SCHEMBL19100596 0.71 KDM4E (0.43) KDM4ETSHRALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538528-A1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089360-A1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed