SCHEMBL19114635

SCHEMBL19114635

Cc1csc(-c2csc(CNC(=O)OC(C)(C)C)n2)n1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.60
HDAC1 Q13547 3/20 0.60
HDAC6 Q9UBN7 3/20 0.60
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
HSP90AA1 P07900 1/20 0.39
PPARA Q07869 2/20 0.39
PI4KB Q9UBF8 1/20 0.38
KDM4A O75164 1/20 0.37
SREBF2 Q12772 1/20 0.37
BACE1 P56817 2/20 0.37
CTSD P07339 1/20 0.37
BACE2 Q9Y5Z0 1/20 0.37
ADORA2A P29274 3/20 0.36
ADORA1 P30542 2/20 0.36
DYRK1A Q13627 1/20 0.36
TGFBR1 P36897 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16020352 0.88 HDAC3 (0.48) HDAC3HDAC1HDAC6NPC1RAB9A
SCHEMBL20691496 0.86 HDAC3 (0.66) HDAC3HDAC1HDAC6SREBF2
SCHEMBL21812678 0.79 MAPK1 (0.53) HDAC3HDAC1HDAC6NPC1RAB9A
SCHEMBL31147895 0.78 HDAC3 (0.49) HDAC3HDAC1HDAC6KDM4A
SCHEMBL21812750 0.78 HDAC3 (0.50) HDAC3HDAC1HDAC6NPC1RAB9A
SCHEMBL21834564 0.78 HDAC3 (0.48) HDAC3HDAC1HDAC6PI4KBKDM4A
SCHEMBL21812752 0.78 HDAC3 (0.48) HDAC3HDAC1HDAC6PI4KBKDM4A
SCHEMBL215719 0.78 HDAC3 (0.51) HDAC3HDAC1HDAC6KDM4A
SCHEMBL21812652 0.77 LMNA (0.53) HDAC3HDAC1HDAC6NPC1RAB9A
SCHEMBL21812758 0.77 HDAC3 (0.49) HDAC3HDAC1HDAC6NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2708534-B1 THIAZOLE COMPOUND AND PREPARATION METHOD AND USE THEREOF SHANGHAI THEORION PHARMACEUTICAL CO LTD (CN) 2017-07-12 EP disclosed