SCHEMBL21812752

SCHEMBL21812752

Cc1nc(-c2csc(CNC(=O)OC(C)(C)C)n2)n[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.48
HDAC6 Q9UBN7 4/20 0.48
HDAC1 Q13547 3/20 0.48
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
GFER P55789 3/20 0.37
CYP1A2 P05177 1/20 0.37
NCOR2 Q9Y618 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
PTPRB P23467 1/20 0.35
KDM4A O75164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPK1 P28482 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21834564 0.80 HDAC3 (0.48) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL21812678 0.79 MAPK1 (0.53) HDAC3HDAC6HDAC1LMNAPTPRB
SCHEMBL21812888 0.78 RAB9A (0.49) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL21812556 0.78 HDAC3 (0.48) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL19114635 0.78 HDAC3 (0.60) HDAC3HDAC6HDAC1PI4KBKDM4A
SCHEMBL21812750 0.78 HDAC3 (0.50) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL16020352 0.78 HDAC3 (0.48) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL21812652 0.77 LMNA (0.53) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL21812758 0.77 HDAC3 (0.49) HDAC3HDAC6HDAC1KDM4ELMNA
SCHEMBL21812580 0.75 HDAC3 (0.50) HDAC3HDAC6HDAC1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020064175-A1 INDANE DERIVATIVES FOR USE IN THE TREATMENT OF BACTERIAL INFECTION ANTABIO SAS (FR) 2020-04-02 WO disclosed
EP-3628672-A1 INDANE DERIVATIVES FOR USE IN THE TREATMENT OF BACTERIAL INFECTION Antabio SAS (FR) 2020-04-01 EP disclosed