SCHEMBL19132829

SCHEMBL19132829

CCC1(C)CCC(NC(=O)c2cn[nH]c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.41
ROCK2 O75116 4/20 0.39
ROCK1 Q13464 2/20 0.39
HPGDS O60760 1/20 0.39
CD38 P28907 1/20 0.38
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38
SMYD3 Q9H7B4 1/20 0.38
AR P10275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1609860 0.81 CD38 (0.47) ROCK2ROCK1CD38SMYD3
SCHEMBL4886377 0.78 SMN1; SMN2 (0.51) ROCK2
SCHEMBL19132785 0.78 RORC (0.48) RORCHPGDSAR
SCHEMBL19132740 0.76 ROCK2 (0.40) RORCROCK2ROCK1HPGDSCD38
SCHEMBL20387472 0.76 SMYD3 (0.54) HPGDSSMYD3
SCHEMBL11898543 0.75 HPGDS (0.48) ROCK2ROCK1HPGDSKDM1A
SCHEMBL19132783 0.73 RORC (0.51) RORCHPGDSSMYD3
SCHEMBL19139056 0.71 RORC (0.50) RORC
SCHEMBL19132827 0.70 TSHR (0.45) RORC
SCHEMBL24767228 0.70 EPHX2 (0.40) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9708253-B2 Cyclohexyl sulfone RORγ modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2017-07-18 US disclosed