SCHEMBL19159014

SCHEMBL19159014

Cc1nc(Oc2cccc(F)c2F)nc2cnccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 2/20 0.40
F3 P13726 2/20 0.40
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
HTR1A P08908 1/20 0.39
DHODH Q02127 2/20 0.38
F10 P00742 1/20 0.36
TRPA1 O75762 1/20 0.36
CXCR2 P25025 1/20 0.36
MAPK1 P28482 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
KDM4C Q9H3R0 4/20 0.35
PIP4K2A P48426 1/20 0.35
LATS1 O95835 1/20 0.34
SLC6A3 Q01959 1/20 0.34
ALDH1A1 P00352 1/20 0.33
ESR1 P03372 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
FFAR1 O14842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17503821 0.85 F7 (0.40) F7F3SLC6A2SLC6A4HTR1A
SCHEMBL19158869 0.79 HTT (0.40) KDM4CLATS1
SCHEMBL19158876 0.75 KDM4C (0.41) KDM4CLATS1
SCHEMBL17503670 0.74 MAPK1 (0.42) F7F3DHODHF10MAPK1
SCHEMBL19159348 0.73 ALDH1A1 (0.41) KDM4CLATS1ALDH1A1
SCHEMBL19158957 0.72 CXCR2 (0.44) F7F3DHODHF10CXCR2
SCHEMBL19158797 0.72 PTGS1 (0.46) MAPK1KDM4CALDH1A1
SCHEMBL19159015 0.72 CXCR2 (0.44) F7F3DHODHF10CXCR2
SCHEMBL19158281 0.69 KDM4C (0.51) KDM4CPIP4K2ALATS1
SCHEMBL19158774 0.69 KDM4C (0.39) KDM4CLATS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970211-B1 HISTONE DEMETHYLASE INHIBITORS QUANTICEL PHARMACEUTICALS INC (US) 2017-07-26 EP disclosed