SCHEMBL19159686

SCHEMBL19159686

O=C(c1cccnc1)N1CCC2(CC2)C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.62
VNN1 O95497 1/20 0.55
BTD P43251 1/20 0.55
ALDH1A1 P00352 1/20 0.54
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.53
PKM P14618 1/20 0.53
MAPK1 P28482 1/20 0.53
POLB P06746 1/20 0.52
SPR P35270 1/20 0.52
CHRNB2 P17787 1/20 0.51
CHRNB4 P30926 1/20 0.51
CHRNA3 P32297 1/20 0.51
CHRNA7 P36544 1/20 0.51
CHRNA4 P43681 1/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
CYP3A4 P08684 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17444269 0.86 OPRM1 (0.58) CHRM2VNN1BTDALDH1A1LMNA
SCHEMBL4815807 0.85 MAPK1 (0.57) CHRM2ALDH1A1LMNAHPGDPKM
SCHEMBL4815797 0.85 MAPK1 (0.57) CHRM2ALDH1A1LMNAHPGDPKM
SCHEMBL10700296 0.83 CHRM2 (0.57) CHRM2ALDH1A1LMNAPKMMAPK1
SCHEMBL19159945 0.83 CYP3A4 (0.68) ALDH1A1HPGDMEN1KMT2ACYP3A4
SCHEMBL17443920 0.82 OPRM1 (0.48) CHRM2VNN1BTDALDH1A1LMNA
SCHEMBL5446400 0.82 CHRM2 (0.65) CHRM2ALDH1A1LMNAPKMMAPK1
SCHEMBL14731514 0.82 MAPK1 (0.53) CHRM2ALDH1A1LMNAHPGDPKM
SCHEMBL17444174 0.82 CHRM2 (0.45) CHRM2VNN1BTDALDH1A1LMNA
SCHEMBL19159719 0.81 MGLL (0.66) CHRM2ALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3196199-A2 SUBSTITUTED N-(PYRROLIDINE-3-YL)-7H-PYRROLO[2,3-D]PYRIMIDINE-4-AMINE AS JANUS KINASE INHIBITOR Yang Ji Chemical Co., Ltd. (KR) 2017-07-26 EP disclosed