SCHEMBL19160331

SCHEMBL19160331

CCc1ccn(Cc2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.50
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP19A1 P11511 3/20 0.44
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
TBXAS1 P24557 1/20 0.44
QPCT Q16769 1/20 0.44
CYP4Z1 Q86W10 1/20 0.44
QPCTL Q9NXS2 1/20 0.44
SIGMAR1 Q99720 1/20 0.39
MAPK14 Q16539 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28125757 0.85 CYP19A1 (0.46) TP53CA12CA1CA2CA9
SCHEMBL28129581 0.82 CA12 (0.47) CA12CA1CA2CA9CYP2C19
SCHEMBL1733332 0.80 CYP2C19 (0.50) CA12CA1CA2CA9CYP2C19
SCHEMBL1680504 0.80 LOXL2 (0.50) CA12CA1CA2CA9CYP2C19
SCHEMBL28878337 0.79 ALDH1A1 (0.55) CA12CA1CA2CA9CYP2C19
SCHEMBL1564273 0.78 CA12 (0.47) TP53CA12CA1CA2CA9
SCHEMBL27889596 0.77 TDP1 (0.54) CA12CA1CA2CA9CYP2C19
SCHEMBL9435256 0.77 CYP2C19 (0.47) CA12CA1CA2CA9CYP2C19
SCHEMBL1234635 0.77 CYP2C19 (0.44) CA12CA1CA2CA9CYP2C19
SCHEMBL28139247 0.77 CYP2A6 (0.58) CYP19A1MAPTCYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109535164-A JAK kinase inhibitor, preparation method thereof and application thereof in medical field 上海华汇拓医药科技有限公司 2019-03-29 CN disclosed
EP-1921077-B1 AGENT FOR TREATING AND/OR PREVENTING SLEEP DISORDER KYOWA HAKKO KIRIN CO LTD (JP) 2017-07-26 EP disclosed