SCHEMBL9435256

SCHEMBL9435256

O=CCc1ccn(Cc2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
MAPT P10636 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 1/20 0.42
POLB P06746 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
TBXAS1 P24557 1/20 0.42
QPCT Q16769 1/20 0.42
CYP4Z1 Q86W10 1/20 0.42
QPCTL Q9NXS2 1/20 0.42
ALDH1A1 P00352 4/20 0.40
LMNA P02545 4/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28129581 0.79 CA12 (0.47) CYP2C19CA12CA1CA2CA9
SCHEMBL510501 0.78 DRD2 (0.52) CYP2C19CA12CA1CA2CA9
SCHEMBL1733332 0.77 CYP2C19 (0.50) CYP2C19CA12CA1CA2CA9
SCHEMBL1680504 0.77 LOXL2 (0.50) CYP2C19CA12CA1CA2CA9
SCHEMBL19160331 0.77 TP53 (0.50) CYP2C19CA12CA1CA2CA9
SCHEMBL28125757 0.74 CYP19A1 (0.46) CYP2C19CA12CA1CA2CA9
SCHEMBL27889596 0.74 TDP1 (0.54) CYP2C19CA12CA1CA2CA9
SCHEMBL1234635 0.74 CYP2C19 (0.44) CYP2C19CA12CA1CA2CA9
SCHEMBL13515393 0.74 CYP2C19 (0.44) CYP2C19CA12CA1CA2CA9
SCHEMBL10667139 0.73 CYP2C19 (0.43) CYP2C19CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994003446-A1 4-SUBSTITUTED 1,2,4-TRIAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1994-02-17 WO disclosed