Methoxsalen

Methoxsalen

SCHEMBL19168

COc1c2occc2cc2ccc(=O)oc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 1.00
MAOA P21397 3/20 1.00
CYP1A2 P05177 2/20 1.00
CYP2A6 P11509 2/20 1.00
MAPK1 P28482 2/20 1.00
CYP2C19 P33261 2/20 1.00
CYP2D6 P10635 1/20 1.00
TSHR P16473 1/20 1.00
ACHE P22303 1/20 1.00
PDE4A P27815 1/20 1.00
SLC6A3 Q01959 1/20 1.00
CYP2A13 Q16696 1/20 1.00
KDM4E B2RXH2 6/20 0.69
HSD17B10 Q99714 4/20 0.69
POLB P06746 2/20 0.69
MAPT P10636 2/20 0.69
MAOB P27338 1/20 0.65
ALDH1A1 P00352 6/20 0.62
HPGD P15428 5/20 0.62
CA9 Q16790 5/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methoxsalen SCHEMBL2302069 1.00 CYP3A4 (1.00) CYP3A4MAOACYP1A2CYP2A6MAPK1
Methoxsalen SCHEMBL29376525 1.00 CYP3A4 (1.00) CYP3A4MAOACYP1A2CYP2A6MAPK1
Methoxsalen SCHEMBL6142553 0.98 CYP3A4 (0.97) CYP3A4MAOACYP1A2CYP2A6MAPK1
Methoxsalen SCHEMBL9387169 0.93 CYP3A4 (0.86) CYP3A4MAOACYP1A2CYP2A6MAPK1
Methoxsalen SCHEMBL10572509 0.92 CYP3A4 (0.84) CYP3A4MAOACYP1A2CYP2A6MAPK1
Methoxsalen SCHEMBL598765 0.90 CYP3A4 (0.82) CYP3A4MAOACYP1A2CYP2A6MAPK1
Bergapten SCHEMBL9792363 0.86 CYP3A4 (0.74) CYP3A4MAOACYP1A2CYP2A6MAPK1
SCHEMBL7781220 0.84 CYP3A4 (0.72) CYP3A4MAOACYP1A2CYP2A6MAPK1
SCHEMBL18788583 0.83 CYP3A4 (0.71) CYP3A4MAOACYP1A2CYP2A6MAPK1
SCHEMBL13660657 0.83 CYP3A4 (0.71) CYP3A4MAOACYP1A2CYP2A6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 21232 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4007582-B1 ANTIBIOTICS IN COMBINATION WITH PHOTODYNAMIC THERAPY FOR USE IN A METHOD OF ENHANCING THE ANTIMICROBIAL ACTION OF SYSTEMICALLY ADMINISTERED ANTIBIOTICS KOITE HEALTH OY (FI) 2026-05-20 EP claimed
CN-122056865-A Application of xanthotoxin in preparation of medicines for treating liver cancer 蕲春县人民医院 2026-05-19 CN claimed
US-20260131003-A1 Method and kit for treating skin infections KOITE HEALTH OY (FI) 2026-05-14 US claimed
EP-4255560-B1 KIT FOR TREATMENT OF PATIENTS HAVING DRY MOUTH SYNDROME KOITE HEALTH OY (FI) 2026-04-22 EP claimed
US-20260096569-A1 EDIBLE COATING WITH ANTIMICROBIAL PROPERTIES APEEL TECH INC (US) 2026-04-09 US claimed
US-20260061057-A1 METHOD FOR GENERATING IMMUNOREGULATORY CELLS IN A BLOOD-DERIVED SAMPLE THERAKOS DEVELOPMENT LTD (IE) 2026-03-05 US claimed
EP-4680203-A1 COMPOSITIONS FOR SUSTAINED RELEASE OF POORLY SOLUBLE ACTIVE INGREDIENTS Prolevi Bio AB (SE) 2026-01-21 EP claimed
US-12521436-B2 Method and kit for treating skin infections KOITE HEALTH OY (FI) 2026-01-13 US claimed
US-12509465-B2 Benzoimidazole derivatives as anticancer agents CENTRE LEON BERARD (FR) 2025-12-30 US claimed
US-20250388642-A1 COMPOSITIONS AND METHODS FOR IMPROVED NK CELL THERAPIES CERUS CORPORATION (US) 2025-12-25 US claimed
EP-0165313-A1 NUCLEIC ACID HYBRIDIZATION ASSAY. HYDROCARBON RESEARCH INC (US) 1985-12-27 EP claimed
WO-1985002628-A1 NUCLEIC ACID HYBRIDIZATION ASSAY HRI RESEARCH, INC. (US) 1985-06-20 WO claimed
EP-0138489-A1 Apparatus and methods for treating cells with radiation McNeilab, Inc. (US) 1985-04-24 EP claimed
US-4454152-A WITH POLYOXYETHYLENE GLYCOL, FOR ORAL ADMINISTRATION HOFFMANN-LA ROCHE INC. (US) 1984-06-12 US claimed
US-4321919-A Method and system for externally treating human blood LEUKOCYTE RESEARCH, INC. (US) 1982-03-30 US claimed
EP-0039874-A2 Methoxsalen compositions and their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-11-18 EP claimed
US-RE30376-E 8-Methoxypsoralen THOMAS C. ELDER, INC. (US) 1980-08-19 US claimed
US-RE30377-E Process for making ω-chloro-2,3,4-trihydroxyacetophenone THOMAS C. ELDER, INC. (US) 1980-08-19 US claimed
US-4129575-A 8-Methoxypsoralen THOMAS C. ELDER, INC. (US) 1978-12-12 US claimed
US-4129576-A Process for making ω-chloro-2,3,4-trihydroxyacetophenone THOMAS C. ELDER, INC. (US) 1978-12-12 US claimed