SCHEMBL19188055

SCHEMBL19188055

Cc1ccc(-c2ccc3c(c2)NC(=O)CO3)cc1

nearest known ligand 0.77

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.77
KDM4E B2RXH2 4/20 0.62
RAB9A P51151 3/20 0.62
NPC1 O15118 2/20 0.62
MAPT P10636 7/20 0.60
NR3C2 P08235 4/20 0.58
PARP1 P09874 1/20 0.57
ALDH1A1 P00352 3/20 0.56
PDE3B Q13370 1/20 0.55
PDE3A Q14432 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
HPGD P15428 1/20 0.54
DRD2 P14416 1/20 0.54
DRD4 P21917 1/20 0.54
DRD3 P35462 1/20 0.54
KMT2A Q03164 1/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19188092 0.88 MMP12 (0.62) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL279594 0.87 MMP12 (1.00) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL4267366 0.87 MMP12 (0.70) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL304764 0.86 MAPT (0.62) MMP12KDM4EMAPTNR3C2PARP1
SCHEMBL5214057 0.83 ALDH1A1 (0.60) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL4264682 0.81 MMP12 (0.58) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL4267784 0.81 PKM (0.59) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL14423461 0.81 MMP12 (0.54) MMP12KDM4ERAB9ANPC1MAPT
SCHEMBL4271023 0.81 MMP12 (0.70) MMP12RAB9ANR3C2PARP1DRD2
SCHEMBL4259548 0.80 POLB (0.78) MMP12KDM4ERAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2758398-B1 SUBSTITUTED N- [1-CYANO-2- (PHENYL) ETHYL]-2-AZABICYCLO [2.2.1]HEPTANE-3-CARBOXAMIDE INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2017-08-02 EP disclosed