SCHEMBL19190702

SCHEMBL19190702

Cc1cc(-c2cc(F)c(=N)n(C(=N)COc3ccnc4cc(O)ccc34)c2)on1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MET P08581 19/20 0.43
CYP3A4 P08684 2/20 0.31
TLR8 Q9NR97 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2695965 0.77 MET (0.60) MET
SCHEMBL18061173 0.74 MET (0.48) METCYP3A4
SCHEMBL9910476 0.70 MET (0.81) METCYP3A4
Bromide SCHEMBL2699721 0.70 MET (0.79) METCYP3A4
SCHEMBL13772484 0.67 MET (0.49) MET
SCHEMBL19190560 0.66 MET (0.60) MET
SCHEMBL2699919 0.65 MET (0.64) METCYP3A4
SCHEMBL14848256 0.63 MET (0.46) METCYP3A4
SCHEMBL19190876 0.62 MET (0.62) MET
SCHEMBL4299513 0.61 KDM4E (0.43) METTLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2231663-B1 6-([1,2,4]TRIAZOLO[4,3-A]PYRIDIN-3-YLMETHYL)-1,6-NAPHTHYRIDIN-5(6H)-ONE DERIVATIVES AS C-MET INHIBITORS AMGEN INC (US) 2017-08-02 EP disclosed