SCHEMBL19192563

SCHEMBL19192563

C[C@H](NC(=O)OC(C)(C)C)C(=O)NNCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.55
CTSS P25774 5/20 0.50
CTSK P43235 5/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA7 P43166 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
PPARA Q07869 2/20 0.49
KMT2A Q03164 1/20 0.48
BACE1 P56817 3/20 0.48
PPARG P37231 1/20 0.46
SYK P43405 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29253632 0.86 BACE1 (0.59) ATMCTSSCTSKCA12CA1
SCHEMBL30279569 0.86 BACE1 (0.59) ATMCTSSCTSKCA12CA1
SCHEMBL2393583 0.86 BACE1 (0.59) ATMCTSSCTSKCA12CA1
SCHEMBL24347009 0.84 BACE1 (0.60) ATMCTSSCTSKCTSLCTSB
SCHEMBL5738490 0.83 CTSS (0.51) ATMCTSSCTSKCTSLCTSB
SCHEMBL4212585 0.83 CTSK (0.62) ATMCTSSCTSKCTSLCTSB
SCHEMBL4632779 0.83 CA12 (0.60) ATMCTSSCTSKCA12CA1
SCHEMBL6842587 0.82 CTSS (0.53) ATMCTSSCTSKCTSLCTSB
SCHEMBL7984152 0.82 CTSS (0.53) ATMCTSSCTSKCTSLCTSB
SCHEMBL6842589 0.82 CTSS (0.53) ATMCTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2771337-B1 3-(PYRIMIDIN-4-YL)-OXAZOLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2017-08-02 EP disclosed