SCHEMBL19193000

SCHEMBL19193000

COc1ccc2c(c1)c(CC#N)cn2C

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.63
HTR6 P50406 3/20 0.60
MTNR1A P48039 9/20 0.54
MTNR1B P49286 9/20 0.54
NQO2 P16083 1/20 0.54
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7496635 0.88 ALDH1A1 (0.51) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL13888101 0.81 ADRB2 (0.70) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL1093061 0.81 ADRB2 (0.65) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL14041509 0.80 HTR6 (0.48) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL2726199 0.80 AKR1C3 (0.66) HTR6MTNR1AMTNR1BNQO2RAB9A
SCHEMBL12185393 0.79 ADRB2 (0.76) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL6261747 0.79 ADRB2 (0.67) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL10577553 0.79 ADRB2 (0.44) ADRB2HTR6MTNR1AMTNR1BNQO2
SCHEMBL6245487 0.79 CYP2A6 (0.48) ADRB2HTR6MEN1POLBRAB9A
SCHEMBL13015284 0.79 ALDH1A1 (0.49) ADRB2HTR6MEN1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445497-B1 Use of derivatives of indoles for the treatment of cancer CENTRE NAT DE LA RECH SCIENT (C N R S ) (FR) 2017-08-02 EP disclosed