SCHEMBL19200534

SCHEMBL19200534

COC(=O)C(c1ccc(F)cc1F)N1CCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
KMT2A Q03164 1/20 0.49
NR3C2 P08235 4/20 0.45
NPY2R P49146 1/20 0.41
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
SLC6A2 P23975 2/20 0.40
NR3C1 P04150 1/20 0.39
OPRM1 P35372 2/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 1/20 0.39
RAB9A P51151 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19200535 0.86 CES2 (0.40) MEN1ALDH1A1LMNAKMT2ANR3C2
SCHEMBL20696322 0.86 CES2 (0.40) MEN1ALDH1A1LMNAKMT2ANPY2R
SCHEMBL19182797 0.84 LMNA (0.45) LMNANPY2RCES2CES1SLC6A2
SCHEMBL15063187 0.79 GAA (0.50) MEN1ALDH1A1LMNAKMT2ANPY2R
SCHEMBL31560789 0.79 CES2 (0.46) ALDH1A1NR3C2CES2CES1RAB9A
SCHEMBL31117167 0.79 CES2 (0.46) ALDH1A1NR3C2CES2CES1RAB9A
SCHEMBL15797720 0.78 CHRNB2 (0.42) MEN1ALDH1A1KMT2ANPY2RCES2
SCHEMBL15063231 0.77 LMNA (0.71) MEN1ALDH1A1LMNAKMT2ANR3C2
SCHEMBL8595608 0.75 CES2 (0.58) LMNANR3C2CES2CES1RAB9A
SCHEMBL6400373 0.75 CES2 (0.58) LMNANR3C2CES2CES1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017131221-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-03 WO disclosed