SCHEMBL19202358

SCHEMBL19202358

COc1ccc(C2CNC2)c(Cl)c1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.54
CHRNA4 P43681 4/20 0.54
CHRNB4 P30926 1/20 0.54
CHRNA3 P32297 1/20 0.54
CHRNA7 P36544 1/20 0.54
HTR2C P28335 6/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HTR2A P28223 3/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22324792 0.83 HTR2C (0.58) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL28706083 0.79 NSD2 (0.49)
SCHEMBL18117756 0.79 MTNR1A (0.64) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL19559348 0.79 MTNR1A (0.64) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL28713145 0.78 TAS1R3 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL28710470 0.77 TAS1R3 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL20010694 0.76 TAS1R3 (0.43)
SCHEMBL9820701 0.74 SLC6A2 (0.51) HTR2CSLC6A2SLC6A4SLC6A3
SCHEMBL1437913 0.74 NPC1 (0.43)
SCHEMBL28694993 0.73 TAS1R3 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128896-A1 FXR AGONIST AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2017-08-03 WO disclosed