SCHEMBL19202540

SCHEMBL19202540

COc1ccc(C2(O)CN(C(=O)OC(C)(C)C)C2)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
STS P08842 2/20 0.42
MET P08581 1/20 0.41
AXL P30530 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
ESR2 Q92731 1/20 0.40
ROCK2 O75116 1/20 0.39
EPHX2 P34913 1/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
CTSD P07339 1/20 0.39
CTSE P14091 1/20 0.39
BACE1 P56817 1/20 0.39
SLC2A1 P11166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19689482 0.85 MET (0.37) ALDH1A1STSMETAXLGPR119
SCHEMBL29736070 0.85 MET (0.37) ALDH1A1STSMETAXLGPR119
SCHEMBL29735795 0.85 ESR2 (0.53) STSMETAXLESR2MEN1
SCHEMBL19689567 0.85 ESR2 (0.53) STSMETAXLESR2MEN1
SCHEMBL30148531 0.84 STS (0.50) ALDH1A1STSMETAXLGPR119
SCHEMBL31735017 0.84 RORC (0.42) ALDH1A1STSESR2ROCK2MEN1
SCHEMBL30148522 0.84 STS (0.50) ALDH1A1STSMETAXLGPR119
SCHEMBL15689748 0.81 STS (0.44) STSGPR119ESR2MAPTMEN1
SCHEMBL29853675 0.80 CYP3A4 (0.40) ALDH1A1STSMETAXLGPR119
SCHEMBL26768529 0.80 CYP3A4 (0.40) ALDH1A1STSMETAXLGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128896-A1 FXR AGONIST AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2017-08-03 WO disclosed