SCHEMBL19202545

SCHEMBL19202545

COC(=O)c1cn(C2CC2)c2cc(Br)ccc12

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PRPS1 P60891 2/20 0.51
NR4A2 P43354 4/20 0.43
KRAS P01116 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
CHEK1 O14757 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CG P48736 1/20 0.39
ALDH1A1 P00352 3/20 0.39
GAA P10253 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
THRB P10828 1/20 0.39
MAPK8 P45983 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2592735 0.82 PRPS1 (0.39) PRPS1NR4A2L3MBTL1
SCHEMBL497718 0.79 NR4A2 (0.63) PRPS1NR4A2KMT2AMEN1L3MBTL1
SCHEMBL7512469 0.78 LMNA (0.58) KMT2AMEN1PIK3CDPIK3R1PIK3CA
SCHEMBL29576838 0.78 LMNA (0.58) KMT2AMEN1PIK3CDPIK3R1PIK3CA
SCHEMBL29576694 0.77 KDM4E (0.59) KMT2AMEN1PIK3CDPIK3R1PIK3CA
SCHEMBL7578838 0.77 KDM4E (0.59) KMT2AMEN1PIK3CDPIK3R1PIK3CA
SCHEMBL2596068 0.77 OPRK1 (0.42) PRPS1ALDH1A1GAASMN1; SMN2
SCHEMBL498716 0.76 PRPS1 (0.45) PRPS1NR4A2KRASKMT2AMEN1
SCHEMBL21549969 0.76 NR4A2 (0.66) PRPS1NR4A2KRASKMT2AMEN1
SCHEMBL35211208 0.76 NR4A2 (0.66) PRPS1NR4A2KRASKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128896-A1 FXR AGONIST AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2017-08-03 WO disclosed