SCHEMBL19205359

SCHEMBL19205359

c1ccc(C2CCCC2)c(OC[C@H]2CCNC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 10/20 0.52
SLC6A4 P31645 10/20 0.52
HTR1A P08908 8/20 0.52
SLC6A3 Q01959 6/20 0.52
PTGDR2 Q9Y5Y4 1/20 0.49
HTR2C P28335 3/20 0.48
HTR1D P28221 2/20 0.45
HTR1B P28222 2/20 0.45
CYP1A2 P05177 2/20 0.43
ADRA2A P08913 2/20 0.43
CYP2D6 P10635 2/20 0.43
ADRA1A P35348 2/20 0.43
THRB P10828 1/20 0.43
TSHR P16473 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1D P25100 1/20 0.43
CYP2C19 P33261 1/20 0.43
ADRA1B P35368 1/20 0.43
THPO P40225 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19205356 1.00 SLC6A2 (0.52) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
SCHEMBL19205318 1.00 SLC6A2 (0.52) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
SCHEMBL19240459 0.99 SLC6A2 (0.51) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
Hydrochloric Acid SCHEMBL19205314 0.97 SLC6A2 (0.50) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
Hydrochloric Acid SCHEMBL19205459 0.97 SLC6A2 (0.50) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
SCHEMBL19240458 0.97 SLC6A2 (0.52) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
Hydrochloric Acid SCHEMBL19205346 0.96 SLC6A2 (0.51) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
Hydrochloric Acid SCHEMBL19205397 0.96 SLC6A2 (0.51) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
SCHEMBL5801431 0.84 SLC6A2 (0.61) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2
Hydrochloric Acid SCHEMBL19205421 0.83 SLC6A2 (0.55) SLC6A2SLC6A4HTR1ASLC6A3PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3210971-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2019-10-16 EP disclosed
US-9944596-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-17 US disclosed
US-9944596-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-04-17 US disclosed
EP-3210971-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2017-08-30 EP disclosed
US-20170233339-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-17 US disclosed
US-20170233339-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-17 US disclosed
US-20170233339-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233339-A1 HETEROCYCLIC COMPOUND RBP4, RBP1, RARA SLC6A2 4083/4885SLC6A4 2662/4885HTR1A 4037/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.