SCHEMBL1920570

SCHEMBL1920570

CCCNC(=O)c1nc[nH]n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.42
LMNA P02545 2/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.39
TDP1 Q9NUW8 2/20 0.38
THRB P10828 1/20 0.38
RECQL P46063 1/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38
DPP4 P27487 2/20 0.38
RIPK1 Q13546 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10245160 0.90 TSHR (0.49) L3MBTL1KDM4ESMN1; SMN2MMP2NPC1
SCHEMBL13263618 0.88 NAAA (0.49) LMNAL3MBTL1KDM4ESMN1; SMN2NPC1
SCHEMBL1763316 0.87 CCNE2 (0.39) LMNARIPK1SMN1; SMN2NPC1RAB9A
SCHEMBL10780680 0.87 NAAA (0.51) LMNAL3MBTL1KDM4ESMN1; SMN2
SCHEMBL22372109 0.84 KDM4E (0.48) KDM4EKMT2ASMN1; SMN2TP53
SCHEMBL30162712 0.84 ACR (0.40) POLBL3MBTL1KDM4EKMT2ARAB9A
SCHEMBL9999597 0.82 MAOB (0.45) LMNAKDM4EKMT2A
SCHEMBL31469580 0.81 HTT (0.49) LMNAGAAKMT2ASMN1; SMN2NPC1
SCHEMBL27921654 0.81 LMNA (0.41) LMNAL3MBTL1KDM4EKMT2ANPSR1
SCHEMBL19852903 0.79 MAPK8 (0.42) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326181-A1 ANTIFUNGAL AGENTS Merck Sharp & Dohme Corp. (US) 2011-06-01 EP disclosed
WO-2010019204-A1 ANTIFUNGAL AGENTS MERCK SHARP & DOHME CORP. (US) 2010-02-18 WO disclosed
EP-0126326-B1 PROCESS FOR PREPARING 1,2,4-TRIAZOLE-3-CARBOXAMIDES UBE INDUSTRIES, LTD. (JP) 1987-08-05 EP disclosed
US-4578479-A Process for preparing 1,2,4-triazole-3-carboxamides UBE INDUSTRIES, LTD. (JP) 1986-03-25 US disclosed
EP-0126326-A1 Process for preparing 1,2,4-triazole-3-carboxamides UBE INDUSTRIES, LTD. (JP) 1984-11-28 EP disclosed