SCHEMBL19209593

SCHEMBL19209593

FC(F)(F)c1ccc2c(Nc3ccccc3)cc(C(F)(F)F)nc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.52
MAPT P10636 3/20 0.52
ALDH1A1 P00352 2/20 0.52
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.52
GFER P55789 1/20 0.52
KMT2A Q03164 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
IDH2 P48735 1/20 0.49
TLR7 Q9NYK1 1/20 0.48
ACP1 P24666 2/20 0.46
IGF1R P08069 4/20 0.45
ABCG2 Q9UNQ0 5/20 0.45
C1R P00736 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GAK O14976 1/20 0.43
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
MARK3 P27448 1/20 0.42
KDR P35968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29200458 0.80 GAK (0.64) GAAMAPTALDH1A1KDM4EMEN1
SCHEMBL10038804 0.77 CDK2 (0.45) GAAMAPTALDH1A1KDM4EMEN1
SCHEMBL16404469 0.77 ABCG2 (0.76) ALDH1A1KDM4EMEN1KMT2AABCG2
SCHEMBL3826784 0.73 NT5E (0.54) KDM4EIGF1RC1RPRKD3MAP4K4
SCHEMBL19209591 0.73 CTSD (0.41) GAAMAPTALDH1A1KDM4EMEN1
SCHEMBL3453097 0.73 C1R (0.71) MAPTALDH1A1KDM4EC1RNPSR1
SCHEMBL3850835 0.72 BACE1 (0.45) ALDH1A1KDM4EKMT2A
SCHEMBL11133397 0.72 KDM4E (0.49) GAAKDM4EMEN1KMT2AC1R
SCHEMBL3828474 0.72 BACE1 (0.45) ALDH1A1KDM4EKMT2A
SCHEMBL11829749 0.72 KDM4E (0.41) ALDH1A1KDM4EKMT2AC1RPRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136642-A1 ANTIBIOTIC COMPOSITIONS THE TRUSTEES OF DARTMOUTH COLLEGE (US) 2017-08-10 WO disclosed
WO-2017136642-A1 ANTIBIOTIC COMPOSITIONS THE TRUSTEES OF DARTMOUTH COLLEGE (US) 2017-08-10 WO disclosed