SCHEMBL1920962

SCHEMBL1920962

O=C(O)c1ccc2c(Cc3ccccc3)n(-c3ccncc3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.43
AURKA O14965 1/20 0.43
CSNK1A1 P48729 1/20 0.43
CDK8 P49336 1/20 0.43
NEK2 P51955 1/20 0.43
LIMK1 P53667 1/20 0.43
CDK5 Q00535 1/20 0.43
DYRK1A Q13627 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
CSNK2A2 P19784 10/20 0.43
CSNK2B P67870 9/20 0.43
CSNK2A1 P68400 6/20 0.43
KDM5A P29375 2/20 0.40
KDM2B Q8NHM5 2/20 0.40
KDM4C Q9H3R0 2/20 0.40
KDM5B Q9UGL1 2/20 0.40
HCAR3 P49019 1/20 0.40
IP6K1 Q92551 1/20 0.40
IP6K3 Q96PC2 1/20 0.40
IP6K2 Q9UHH9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921363 0.93 CHEK1 (0.50) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1922389 0.85 ABCG2 (0.41) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1921689 0.83 IP6K1 (0.48) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1922920 0.81 MPO (0.42) MEN1HPGDKMT2AKHK
SCHEMBL1921732 0.80 CSNK2A2 (0.39) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1920560 0.77 TLR7 (0.42) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1921690 0.77 ELANE (0.34) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1923158 0.75 CHEK1 (0.47) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL13984750 0.73 CDK8 (0.38) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1921349 0.73 CHEK1 (0.45) CHEK1AURKACSNK1A1CDK8NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170833-B1 A TRANSITION METAL CATALYZED SYNTHESIS OF 2H-INDAZOLES SANOFI AVENTIS (FR) 2011-06-01 EP claimed