SCHEMBL19209936

SCHEMBL19209936

C1=C(c2cccc(N3CCN(c4cncnc4)CC3)c2)CCOC1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.42
BACE1 P56817 1/20 0.40
KCNH2 Q12809 1/20 0.40
PIK3CA P42336 4/20 0.39
MTOR P42345 1/20 0.39
PIK3CD O00329 3/20 0.39
RPS6KA3 P51812 1/20 0.37
MAPK14 Q16539 1/20 0.35
FABP7 O15540 1/20 0.35
DYRK1A Q13627 2/20 0.35
PIK3CB P42338 2/20 0.35
PIK3CG P48736 2/20 0.35
PIK3R1 P27986 1/20 0.35
CYP11B2 P19099 1/20 0.35
TLR9 Q9NR96 1/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
HTR1D P28221 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209925 0.78 DHFR (0.65) DHFR
SCHEMBL28058221 0.73 BACE1 (0.46) BACE1KCNH2PIK3CAMTORPIK3CD
SCHEMBL30072245 0.70 FABP7 (0.45) BACE1KCNH2PIK3CAPIK3CDMAPK14
SCHEMBL1570328 0.70 FABP7 (0.45) BACE1KCNH2PIK3CAPIK3CDMAPK14
SCHEMBL932928 0.68 PIK3CD (0.45) PIK3CAPIK3CDMAPK14FABP7DYRK1A
SCHEMBL18857842 0.67 MAPK14 (0.47) PIK3CAMTORPIK3CDMAPK14FABP7
SCHEMBL29415412 0.66 DHFR (0.58) DHFRHTR1AHTR7
SCHEMBL27523614 0.66 MAPT (0.53) DHFRKCNH2
SCHEMBL29387046 0.64 HTR7 (0.69) DHFRHTR1AHTR7
SCHEMBL15577956 0.64 HTR7 (0.69) DHFRHTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3411367-A1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS Vyera Pharmaceuticals, LLC (US) 2018-12-12 EP disclosed
WO-2017136556-A1 COMPOSITIONS AND METHODS FOR TREATING INFECTIONS TURING PHARMACEUTICALS LLC (US) 2017-08-10 WO disclosed